SCHEMBL8901453

SCHEMBL8901453

O=C(O)C(Cc1ccc(OCc2nc3ccccc3s2)cc1)=NO

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.61
RAB9A P51151 4/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
MAPK1 P28482 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
ALOX5 P09917 9/20 0.59
EPHX2 P34913 7/20 0.59
KMT2A Q03164 3/20 0.56
ALDH1A1 P00352 2/20 0.54
MAPT P10636 2/20 0.54
MEN1 O00255 1/20 0.54
KDM4E B2RXH2 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
CYP1A2 P05177 1/20 0.48
CYP2C19 P33261 1/20 0.48
CTBP2 P56545 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8901437 1.00 NPC1 (0.61) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
SCHEMBL9429685 0.83 NPC1 (0.65) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
SCHEMBL1746753 0.79 SMN1; SMN2 (0.67) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
SCHEMBL8626714 0.79 NPC1 (0.60) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
SCHEMBL8626737 0.79 NPC1 (0.60) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
SCHEMBL8622668 0.78 NPC1 (0.58) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
SCHEMBL8622647 0.78 NPC1 (0.58) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
SCHEMBL8136532 0.78 NPC1 (0.73) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
SCHEMBL9427796 0.78 NPC1 (0.60) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1
2-(Phenoxymethyl)Benzothiazole SCHEMBL2245843 0.78 NPC1 (1.00) NPC1RAB9ASMN1; SMN2MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997012866-A1 BIS-HETEROARYLYLMETHOXYPHENYLKETONE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1997-04-10 WO disclosed