SCHEMBL8904757

SCHEMBL8904757

C[C@]12CCC(C(=O)O)=CC1=CC[C@@H]1[C@H]2CC[C@]2(C)C(C(=O)c3ccc(F)cc3)CC[C@@H]12

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 13/20 0.67
SRD5A1 P18405 5/20 0.66
ESR1 P03372 1/20 0.47
AR P10275 1/20 0.47
ESR2 Q92731 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8902462 1.00 SRD5A2 (0.67) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL23752478 0.92 SRD5A2 (0.68) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL21068049 0.92 SRD5A2 (0.68) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL2488075 0.92 SRD5A2 (0.68) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL8163286 0.92 SRD5A2 (0.68) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL29655549 0.92 SRD5A2 (0.70) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL8163428 0.92 SRD5A2 (0.70) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL8163423 0.92 SRD5A2 (0.70) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL8904222 0.90 SRD5A2 (0.56) SRD5A2SRD5A1ESR1ARESR2
SCHEMBL8158983 0.89 SRD5A2 (0.65) SRD5A2SRD5A1ESR1ARESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5683995-A 17 substituted acyl-3-carboxy 3,5-diene steroidals as α-reductase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1997-11-04 US claimed
EP-0673251-A4 1995-10-25 EP claimed
EP-0673251-A1 17 SUBSTITUTED ACYL-3-CARBOXY 3,5-DIENE STEROIDALS AS 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1995-09-27 EP claimed
WO-1994011004-A1 17 SUBSTITUTED ACYL-3-CARBOXY 3,5-DIENE STEROIDALS AS 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-05-26 WO claimed
US-5683995-A 17 substituted acyl-3-carboxy 3,5-diene steroidals as α-reductase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1997-11-04 US disclosed
EP-0673251-A4 1995-10-25 EP disclosed
EP-0673251-A1 17 SUBSTITUTED ACYL-3-CARBOXY 3,5-DIENE STEROIDALS AS 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1995-09-27 EP disclosed
WO-1994011004-A1 17 SUBSTITUTED ACYL-3-CARBOXY 3,5-DIENE STEROIDALS AS 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-05-26 WO disclosed