SCHEMBL8905545

SCHEMBL8905545

Cc1ccc2c(c1)CNCC2c1ccc(O)c(O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.59
MAPK1 P28482 2/20 0.56
CYP3A4 P08684 2/20 0.56
ALOX15 P16050 1/20 0.56
TSHR P16473 1/20 0.56
NFKB1 P19838 1/20 0.56
THPO P40225 1/20 0.56
HSD17B10 Q99714 1/20 0.56
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 1/20 0.54
PMP22 Q01453 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
TAAR1 Q96RJ0 1/20 0.54
ADCY5 O95622 1/20 0.51
SLC6A2 P23975 6/20 0.48
SLC6A4 P31645 6/20 0.48
SLC6A3 Q01959 6/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL9132813 0.99 PARP1 (0.58) PARP1MAPK1CYP3A4ALOX15TSHR
Bromide SCHEMBL8904455 0.88 KDM4E (0.56) PARP1MAPK1CYP3A4ALOX15TSHR
Bromide SCHEMBL8905619 0.84 PARP1 (0.60) PARP1MAPK1CYP3A4ALOX15TSHR
Bromide SCHEMBL8904521 0.82 PARP1 (0.54) PARP1MAPK1CYP3A4ALOX15TSHR
SCHEMBL14494799 0.81 PARP1 (0.68) PARP1MAPK1CYP3A4ALOX15TSHR
SCHEMBL11102977 0.81 PARP1 (0.68) PARP1MAPK1CYP3A4ALOX15TSHR
SCHEMBL22461447 0.80 CYP3A4 (0.66) CYP3A4NFKB1THPOHSD17B10KDM4E
Hydrochloric Acid SCHEMBL11799053 0.80 SLC6A4 (0.61) SLC6A2SLC6A4SLC6A3
SCHEMBL9667782 0.79 PARP1 (0.72) PARP1MAPK1CYP3A4ALOX15TSHR
SCHEMBL8905773 0.78 SLC6A2 (0.46) CYP3A4KDM4EALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5623074-A DERIVATIVES OF 7-DIHYDROXYPHENYL-4,5,6,7-TETRAHYDROTHIAZOLO (4,5-C)PYRIDINE WHICH ACT ON DOPAMINE RECEPTORS; NEPHROVASCULAR DILATORS, DIURETICS, SIDE EFFECT REDUCTION YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed