SCHEMBL8914550

SCHEMBL8914550

O=C(Cc1cccnc1)NC(Cc1c[nH]c2ccccc12)C(=O)NCc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 2/20 0.63
TACR1 P25103 10/20 0.59
MMP2 P08253 2/20 0.58
MMP9 P14780 2/20 0.58
MMP8 P22894 2/20 0.58
SSTR1 P30872 1/20 0.54
SSTR3 P32745 1/20 0.54
CYP3A4 P08684 3/20 0.53
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
TP53 P04637 1/20 0.53
CYP1A2 P05177 1/20 0.53
POLB P06746 1/20 0.53
CYP2D6 P10635 1/20 0.53
MAPT P10636 1/20 0.53
CYP2C9 P11712 1/20 0.53
NFKB1 P19838 1/20 0.53
APEX1 P27695 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8914219 0.91 TACR1 (0.59) BRS3TACR1MMP2MMP9MMP8
SCHEMBL9387236 0.88 TACR1 (0.77) BRS3TACR1MMP2MMP9MMP8
Hydrochloric Acid SCHEMBL8895691 0.87 TACR1 (0.76) BRS3TACR1MMP2MMP9MMP8
SCHEMBL8915040 0.86 TACR1 (0.56) TACR1MMP2MMP9MMP8SSTR1
SCHEMBL9262151 0.83 TACR1 (0.61) TACR1CYP3A4KDM4EMEN1ALDH1A1
SCHEMBL9270608 0.83 TACR1 (0.75) TACR1CYP3A4KDM4EMEN1ALDH1A1
SCHEMBL8893006 0.82 TACR1 (0.73) BRS3TACR1MMP2MMP9MMP8
SCHEMBL9265760 0.82 TACR1 (0.61) BRS3TACR1CYP3A4KDM4EMEN1
SCHEMBL9264952 0.82 TACR1 (0.75) TACR1CYP3A4KDM4EMEN1ALDH1A1
SCHEMBL1459290 0.80 ACE (0.65) TACR1SSTR1SSTR3CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994019320-A1 AROMATIC COMPOUNDS, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1994-09-01 WO claimed
US-5674889-A Aromatic compounds, compositions containing them and their use in therapy MERCK, SHARP & DOHME, LTD. (GB) 1997-10-07 US disclosed
WO-1994019320-A1 AROMATIC COMPOUNDS, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1994-09-01 WO disclosed