SCHEMBL8916080

SCHEMBL8916080

CC(C)Nc1nccnc1N1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.42
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916543 0.79 EPHX2 (0.45) HTR2CEPHX2
SCHEMBL2299768 0.77 EPHX2 (0.51) HTR2CEPHX2
SCHEMBL13116668 0.76 HTR2C (0.56) HTR2CEPHX2
Water SCHEMBL8709610 0.76 EPHX2 (0.50) HTR2CEPHX2
SCHEMBL122262 0.73 USP2 (0.55) HTR2CEPHX2
SCHEMBL14385534 0.72 HTR2C (0.40) HTR2CEPHX2
SCHEMBL23561114 0.72 HTR2C (0.49) HTR2CEPHX2
SCHEMBL13116675 0.71 HTR2C (0.42) HTR2CEPHX2
SCHEMBL859700 0.71 HRH4 (0.72)
SCHEMBL8916808 0.71 HTR2C (0.38) HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686610-A Pyridyl piperazine compound PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
US-5599930-A Substituted indoles as anti-AIDS pharmaceuticals THE UPJOHN COMPANY (US) 1997-02-04 US disclosed
WO-1993001181-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS THE UPJOHN COMPANY (US) 1993-01-21 WO disclosed