SCHEMBL8917912

SCHEMBL8917912

N#CN=C(NCCCCCOc1ccc(Cl)cc1)Nc1cccnc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.63
NAMPT P43490 3/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP2D6 P10635 1/20 0.50
CDK2 P24941 1/20 0.45
FLT4 P35916 1/20 0.45
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
CYP1A2 P05177 1/20 0.41
NOTUM Q6P988 1/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
ABCC9 O60706 2/20 0.40
ABCC8 Q09428 2/20 0.40
KCNJ11 Q14654 2/20 0.40
KCNJ8 Q15842 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918194 0.93 IKBKB (0.53) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
Chs-828 SCHEMBL12083293 0.88 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
Chs-828 SCHEMBL810990 0.88 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
Chs-828 SCHEMBL16312347 0.88 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
SCHEMBL8918236 0.88 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
SCHEMBL8917545 0.88 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
Chs-828 SCHEMBL7142976 0.87 IKBKB (0.79) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
Chs-828 SCHEMBL7148798 0.87 IKBKB (0.79) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
SCHEMBL14324370 0.85 IKBKB (0.52) IKBKBNAMPTCYP3A4CYP2C9CYP2C19
SCHEMBL14324372 0.85 IKBKB (0.52) IKBKBNAMPTCYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696140-A FOR TREATMENT OF ASTHMA, ALLERGIES, NERVOUS SYSTEM DISORDERS OR CANCER LEO PHARMACEUTICAL PRODUCTS LTD. (DK) 1997-12-09 US disclosed