SCHEMBL8921773

SCHEMBL8921773

C1=CC=C2NNNC2N=C1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3600587 0.85
SCHEMBL3514393 0.65
Hydrochloric Acid SCHEMBL29771648 0.57
SCHEMBL188021 0.57
SCHEMBL22536543 0.54
SCHEMBL3584063 0.53
SCHEMBL15132060 0.51
SCHEMBL29342710 0.48
SCHEMBL20245049 0.45
SCHEMBL11667726 0.45

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119119189-A Polypeptides having MMP2 inhibitory effect 大正制药株式会社 2024-12-13 CN disclosed
CN-114450294-B Polypeptides having MMP2 inhibitory effect 大正制药株式会社 2024-11-26 CN disclosed
US-20240199692-A1 POLYPEPTIDE HAVING MMP2-INHIBITORY EFFECT TAISHO PHARMACEUTICAL CO., LTD. (JP) 2024-06-20 US disclosed
WO-2023204170-A1 PROPHYLACTIC OR THERAPEUTIC AGENT, FOR LUNG INFLAMMATION AND FIBROSIS, CONTAINING COMPOUND HAVING MMP2 INHIBITORY ACTIVITY AS ACTIVE INGREDIENT 大正製薬株式会社 2023-10-26 WO disclosed
WO-2022234867-A1 SULFONAMIDE HAVING MMP 7-INHIBITING ACTION 大正製薬株式会社 2022-11-10 WO disclosed
EP-4056581-A1 POLYPEPTIDE HAVING MMP2-INHIBITORY EFFECT Taisho Pharmaceutical Co., Ltd. (JP) 2022-09-14 EP disclosed
CN-114450294-A Polypeptide with MMP2 inhibitory effect 大正制药株式会社 2022-05-06 CN disclosed
US-5674879-A Compositions including and methods of using conformationally restricted angiotensin II antagonist G.D. SEARLE & CO. (US) 1997-10-07 US disclosed