SCHEMBL8922394

SCHEMBL8922394

CCCC(C(=O)S)c1cncnc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
HCAR2 Q8TDS4 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
FFAR2 O15552 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7552546 0.84 AKR1C3 (0.48) AKR1C3AKR1C2HCAR2CYP1A2CYP3A4
SCHEMBL8922398 0.76 AKR1C3 (0.33) AKR1C3AKR1C2
SCHEMBL27412443 0.74 AKR1C3 (0.46) AKR1C3AKR1C2HCAR2HDAC3HDAC1
SCHEMBL1808417 0.71 HCAR2 (0.38) HCAR2
SCHEMBL11007947 0.71 CYP11B1 (0.41) LMNA
SCHEMBL2438138 0.70 AKR1C3 (0.42) AKR1C3AKR1C2HCAR2LMNA
SCHEMBL16919626 0.70 CYP19A1 (0.34)
SCHEMBL18885103 0.69 CYP19A1 (0.33)
SCHEMBL11463162 0.68 SLC6A4 (0.45) CYP3A4
SCHEMBL28131366 0.67 CYP19A1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633379-A N-METHYLASPARTIC ACID ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-05-27 US disclosed