SCHEMBL8923453

SCHEMBL8923453

Nc1ccc2c(ccc3nc(N)[nH]c(=O)c32)c1.Nc1nc2ccc3cccc(N)c3c2c(=O)[nH]1

nearest known ligand 0.78

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TYMS P04818 20/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6653500 0.88 TYMS (1.00) TYMS
SCHEMBL6653412 0.87 TYMS (1.00) TYMS
SCHEMBL6649299 0.79 TYMS (1.00) TYMS
SCHEMBL6651319 0.77 TYMS (1.00) TYMS
SCHEMBL6650266 0.77 TYMS (1.00) TYMS
SCHEMBL30589037 0.77 TYMS (1.00) TYMS
SCHEMBL6654365 0.77 TYMS (1.00) TYMS
SCHEMBL11609746 0.76 TYMS (0.75) TYMS
SCHEMBL6653029 0.75 TYMS (0.81) TYMS
SCHEMBL6649167 0.75 TYMS (1.00) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661155-A THYMIDYLATE SYNTHASE INHIBITOR; ADMINISTERING TO THE MAMMAL SUFFERING FROM LEUKEMIA OR TUMOR 2-(5-(((1,2-DIHYDRO-3-METHYL-1-OXOBENZO(F)QUINAZOLINE-9-YL) METHYL)AMINO)-1-OXO-2-ISOINDOLINYL)GLUTARIC ACID OR SALTS GLAXO WELLCOME INC. (US) 1997-08-26 US disclosed