SCHEMBL8925035

SCHEMBL8925035

CCCCC=Cc1cc(Cl)cc(NC(=O)CBr)c1C(=O)OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
ALDH1A1 P00352 4/20 0.35
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
PDE5A O76074 1/20 0.34
MAPT P10636 3/20 0.33
GAA P10253 2/20 0.33
POLB P06746 2/20 0.33
LMNA P02545 1/20 0.32
GLA P06280 1/20 0.32
THRB P10828 1/20 0.32
GALK1 P51570 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
NPC1 O15118 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8925030 1.00 CYP1A2 (0.37) CYP1A2CYP3A4CYP2C19MEN1KMT2A
SCHEMBL8921606 0.79 SMN1; SMN2 (0.38) CYP1A2CYP3A4CYP2C19MEN1KMT2A
SCHEMBL8921279 0.76 MEN1 (0.40) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL8921612 0.76 SMN1; SMN2 (0.37) CYP1A2CYP3A4CYP2C19KMT2AALDH1A1
SCHEMBL8923316 0.76 MEN1 (0.42) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL8922750 0.74 KMT2A (0.40) MEN1KMT2AALDH1A1MAPTGAA
SCHEMBL7416031 0.73 GALK1 (0.40) CYP1A2CYP2C19MEN1KMT2AALDH1A1
SCHEMBL4733777 0.66 KMT2A (0.55) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL28658975 0.65 CNR1 (0.47) CYP3A4KDM4EMAPTFAAH
SCHEMBL28658973 0.65 CNR1 (0.47) CYP3A4KDM4EMAPTFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633379-A N-METHYLASPARTIC ACID ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-05-27 US disclosed
EP-0685466-A1 3-Heteroaliphatyle-and 3-hetero-(aryle)-aliphatyle-2(1H)-quinolone derivatives CIBA-GEIGY AG (CH) 1995-12-06 EP disclosed