SCHEMBL8929386

SCHEMBL8929386

c1cc2c(c(Nc3ncnc4[nH]ccc34)c1)CCCC2

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.62
TTBK1 Q5TCY1 10/20 0.57
TTBK2 Q6IQ55 10/20 0.57
AKT1 P31749 2/20 0.53
AURKA O14965 1/20 0.51
AURKB Q96GD4 1/20 0.51
INCENP Q9NQS7 1/20 0.51
HPGDS O60760 1/20 0.49
TNNI3K Q59H18 1/20 0.44
MKNK1 Q9BUB5 2/20 0.44
MKNK2 Q9HBH9 2/20 0.44
SYK P43405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787013 0.97 EGFR (0.59) EGFRTTBK1TTBK2AKT1AURKA
Hydrochloric Acid SCHEMBL8929628 0.96 EGFR (0.58) EGFRTTBK1TTBK2AKT1AURKA
SCHEMBL8929866 0.79 EGFR (0.51) EGFRTTBK1TTBK2AKT1AURKA
Hydrochloric Acid SCHEMBL8929855 0.78 EGFR (0.50) EGFRTTBK1TTBK2AKT1AURKA
SCHEMBL27460612 0.75 TTBK1 (0.69) EGFRTTBK1TTBK2AKT1AURKA
SCHEMBL1095145 0.72 EGFR (0.57) EGFR
SCHEMBL8976249 0.72 EGFR (0.65) EGFRMKNK1
SCHEMBL27930913 0.72 TTBK1 (0.64) EGFRTTBK1TTBK2AKT1AURKA
SCHEMBL12101466 0.72 MEN1 (0.56) EGFR
SCHEMBL8929392 0.72 EGFR (0.58) EGFRTTBK1TTBK2AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP claimed
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP disclosed