SCHEMBL8933604

SCHEMBL8933604

CCOC(=O)Oc1c(C)nc2n1-c1ccc(C(C)=O)cc1C(c1ccccc1F)=NC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTAFR P25105 8/20 0.43
GABRA3 P34903 2/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA1 P14867 2/20 0.41
GABRA5 P31644 2/20 0.41
GABRA2 P47869 2/20 0.41
GABRB2 P47870 2/20 0.41
CYP3A4 P08684 2/20 0.41
DRD3 P35462 2/20 0.41
OPRK1 P41145 2/20 0.41
SLC22A1 O15245 1/20 0.41
ABCB11 O95342 1/20 0.41
PDE4D Q08499 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.38
TP53 P04637 1/20 0.36
HTR1A P08908 1/20 0.36
HTR3A P46098 1/20 0.36
KCNH2 Q12809 1/20 0.36
GHSR Q92847 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8933551 0.90 PTAFR (0.46) PTAFRGABRA3GABRG2GABRB3GABRA1
SCHEMBL8933504 0.84 PTAFR (0.50) PTAFRGABRA3GABRG2GABRB3GABRA1
Hydrochloric Acid SCHEMBL8933564 0.83 PTAFR (0.49) PTAFRGABRA3GABRG2GABRB3GABRA1
SCHEMBL8933549 0.81 PTAFR (0.48) PTAFRGABRA3GABRG2GABRB3GABRA1
Hydrochloric Acid SCHEMBL8933661 0.77 PTAFR (0.42) PTAFRGABRA3GABRG2GABRB3GABRA1
SCHEMBL8933501 0.76 PTAFR (0.50) PTAFRGABRA3GABRG2GABRB3GABRA1
SCHEMBL8933595 0.75 PTAFR (0.44) PTAFRGABRA3GABRG2GABRB3GABRA1
SCHEMBL8933412 0.74 PTAFR (0.45) PTAFRGABRA3GABRG2GABRB3GABRA1
SCHEMBL8933546 0.74 CYP3A4 (0.49) PTAFRGABRA3GABRG2GABRB3GABRA1
Hydrochloric Acid SCHEMBL8933629 0.74 PTAFR (0.43) PTAFRGABRA3GABRG2GABRB3GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996023790-A1 ACETYLIMIDAZOBENZODIAZEPINES F. HOFFMANN-LA ROCHE AG (CH) 1996-08-08 WO disclosed