SCHEMBL8936445

SCHEMBL8936445

Cc1cc2c(-c3c(C)cccc3C)c(NC(=O)N(C)Cc3ccccc3)n(C)c(=O)c2cc1C

nearest known ligand 0.83

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 15/20 0.83
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
ABCC1 P33527 1/20 0.42
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936537 0.92 TACR1 (0.78) TACR1CA12CA1CA2CA9
SCHEMBL8936475 0.91 TACR1 (1.00) TACR1TP53
SCHEMBL8936477 0.86 TACR1 (0.77) TACR1TP53
SCHEMBL8936457 0.84 TACR1 (1.00) TACR1
SCHEMBL8936516 0.82 TACR1 (0.77) TACR1
SCHEMBL8784911 0.82 TACR1 (0.68) TACR1TP53
SCHEMBL8936559 0.81 TACR1 (0.90) TACR1
SCHEMBL8936479 0.80 TACR1 (1.00) TACR1CA12CA1CA2CA9
SCHEMBL8936548 0.78 TACR1 (1.00) TACR1TP53
SCHEMBL8936495 0.78 TACR1 (1.00) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5523305-A ANALGESICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-04 US disclosed
EP-0566069-A1 Tachykinin receptor antagonists, isoquinolones and their production TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-20 EP disclosed