SCHEMBL8936576

SCHEMBL8936576

Cc1cc2c(-c3ccccc3)c(NC(=O)NCc3ccccc3)n(C)c(=O)c2cc1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 1.00
ADORA3 P0DMS8 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936527 0.95 TACR1 (0.90) TACR1SMN1; SMN2KDM4EMEN1ALDH1A1
SCHEMBL8936542 0.93 TACR1 (0.86) TACR1SMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL8936454 0.93 TACR1 (0.86) TACR1MEN1ALDH1A1CYP2C19KMT2A
SCHEMBL8936439 0.93 TACR1 (0.86) TACR1SMN1; SMN2MEN1KMT2A
SCHEMBL8936481 0.93 TACR1 (0.86) TACR1SMN1; SMN2KDM4EMEN1HPGD
SCHEMBL8936574 0.91 TACR1 (0.83) TACR1KDM4EMEN1ALDH1A1KMT2A
SCHEMBL8936543 0.89 TACR1 (0.80) TACR1MEN1ALDH1A1KMT2A
SCHEMBL8936580 0.89 TACR1 (0.80) TACR1MEN1ALDH1A1KMT2A
SCHEMBL8936598 0.88 TACR1 (0.78) TACR1
SCHEMBL8936536 0.87 TACR1 (0.77) TACR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5523305-A ANALGESICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-04 US disclosed
EP-0566069-A1 Tachykinin receptor antagonists, isoquinolones and their production TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-20 EP disclosed