SCHEMBL8937659

SCHEMBL8937659

CCOC(=O)C=Cc1cc(Cl)ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.53
ALDH1A1 P00352 3/20 0.53
TTR P02766 1/20 0.49
DPP4 P27487 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49
CYP3A4 P08684 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ESR1 P03372 1/20 0.45
MAOB P27338 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
FDPS P14324 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8937654 1.00 MAPT (0.53) MAPTALDH1A1TTRDPP4CA12
Ethyl 3-(2,4-Dichlorophenyl)Acrylate SCHEMBL1895653 0.88 MAPT (0.58) MAPTALDH1A1TTRDPP4CA12
SCHEMBL31462827 0.88 MAPT (0.50) MAPTALDH1A1TTRDPP4CA12
Ethyl 3-(2,4-Dichlorophenyl)Acrylate SCHEMBL1895655 0.88 MAPT (0.58) MAPTALDH1A1TTRDPP4CA12
SCHEMBL30087204 0.87 MAPT (0.47) MAPTALDH1A1TTRDPP4CA12
SCHEMBL29170149 0.87 MAPT (0.47) MAPTALDH1A1TTRDPP4CA12
SCHEMBL28283048 0.87 TTR (0.58) MAPTALDH1A1TTRDPP4CA12
SCHEMBL31462784 0.87 MAPT (0.49) MAPTALDH1A1TTRDPP4CA12
SCHEMBL28283049 0.87 TTR (0.58) MAPTALDH1A1TTRDPP4CA12
SCHEMBL7922171 0.86 MAPT (0.46) MAPTALDH1A1TTRDPP4CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559109-A Method of treating a PAF-mediated pathology or for treating or preventing psoriasis, nephritis, asthma or shock by administering a PAF antagonist SANKKO COMPANY, LIMITED (JP) 1996-09-24 US disclosed
US-5556852-A PLATELET ACTIVATING FACTOR ANTAGONISTS SANKYO COMPANY, LIMITED (JP) 1996-09-17 US disclosed
US-5369106-A N-acryloylpiperazine derivatives, their preparation and their use of PAF antagonists SANKYO COMPANY, LIMITED (JP) 1994-11-29 US disclosed
US-5192766-A Platelet activating factor antagonist SANKYO COMPANY, LIMITED (JP) 1993-03-09 US disclosed