SCHEMBL8938696

SCHEMBL8938696

Cc1cc(Cl)cc(CN2CCC(Oc3cc4cc[nH]c(=O)c4cc3Cl)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 2/20 0.53
ROCK1 Q13464 2/20 0.43
SCN8A Q9UQD0 4/20 0.42
SCN1A P35498 2/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
ROCK2 O75116 2/20 0.39
PRKACA P17612 4/20 0.39
PRKCD Q05655 1/20 0.39
PRKG1 Q13976 1/20 0.39
PKN1 Q16512 1/20 0.39
PKN2 Q16513 1/20 0.39
AAK1 Q2M2I8 1/20 0.39
CDC42BPA Q5VT25 1/20 0.39
Q6ZSR9 Q6ZSR9 1/20 0.39
BMP2K Q9NSY1 1/20 0.39
CDC42BPB Q9Y5S2 1/20 0.39
PRKACG P22612 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8934996 0.93 MAP2K1 (0.58) MAP2K1ROCK1SCN8ASCN1AMAOA
SCHEMBL8939144 0.93 ROCK1 (0.52) MAP2K1ROCK1SCN8ASCN1AMEN1
SCHEMBL8935003 0.91 MAP2K1 (0.57) MAP2K1ROCK1SCN8ASCN1AMAOA
SCHEMBL8938144 0.89 MAP2K1 (0.53) MAP2K1ROCK1SCN8ASCN1AMAOA
SCHEMBL8938278 0.88 MAP2K1 (0.59) MAP2K1ROCK1SCN8ASCN1AMAOA
SCHEMBL8937925 0.88 ROCK1 (0.54) MAP2K1ROCK1MAOAMAOBROCK2
SCHEMBL8938119 0.87 MAP2K1 (0.55) MAP2K1SCN8ASCN1AMAOAMAOB
SCHEMBL8938641 0.87 ROCK1 (0.54) ROCK1MEN1KMT2AMAOAMAOB
SCHEMBL8938150 0.87 MAP2K1 (0.57) MAP2K1ROCK1MEN1KMT2AMAOA
SCHEMBL8934981 0.86 MAP2K1 (0.59) MAP2K1ROCK1SCN8ASCN1AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed