SCHEMBL8940663

SCHEMBL8940663

COc1c(N2CC3CC3(N)C2)c(F)cc2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.67
KDM4E B2RXH2 9/20 0.65
ALDH1A1 P00352 5/20 0.65
HPGD P15428 4/20 0.65
POLB P06746 3/20 0.65
HSD17B10 Q99714 2/20 0.65
TDP1 Q9NUW8 2/20 0.65
OPRM1 P35372 2/20 0.65
PRKD3 O94806 1/20 0.65
ALOX15 P16050 1/20 0.65
CLK2 P49760 1/20 0.65
CLK4 Q9HAZ1 1/20 0.65
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
LMNA P02545 2/20 0.59
CYP2C19 P33261 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
NPSR1 Q6W5P4 1/20 0.54
ATM Q13315 1/20 0.52
CHRM2 P08172 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28391101 0.92 KCNH2 (0.63) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL30415810 0.92 KCNH2 (0.63) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL8383857 0.90 KCNH2 (0.57) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL6948985 0.90 CYP3A4 (0.58) KCNH2KDM4EALDH1A1HPGDPOLB
Trifluoroacetic Acid SCHEMBL8388928 0.89 KCNH2 (0.61) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL8854414 0.88 KDM4E (0.65) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL9185212 0.87 KCNH2 (0.69) KCNH2KDM4EALDH1A1HPGDPOLB
Hydrochloric Acid SCHEMBL6505726 0.86 KCNH2 (0.72) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL4749958 0.86 KCNH2 (0.60) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL6948982 0.86 KCNH2 (0.49) KCNH2KDM4EALDH1A1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-8048629-A None JP disclosed
JP-H0848629-A PYRIDONECARBOXYLIC ACID DERIVATIVE AND ANTI-PYLORI AGENT WITH THE SAME AS ACTIVE INGREDIENT DAINIPPON PHARMACEUT CO LTD 1996-02-20 JP disclosed