SCHEMBL8941787

SCHEMBL8941787

c1ccc2c(c1)CCc1cc(C3CO3)ccc1-2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
SRD5A1 P18405 1/20 0.45
SRD5A2 P31213 1/20 0.45
RAB9A P51151 3/20 0.41
NPC1 O15118 3/20 0.41
CES1 P23141 1/20 0.39
MITF O75030 1/20 0.39
HSP90AA1 P07900 1/20 0.39
PARP1 P09874 1/20 0.37
SETD7 Q8WTS6 1/20 0.36
NR1H2 P55055 2/20 0.35
NR1H3 Q13133 2/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 4/20 0.35
MAPT P10636 4/20 0.35
HPGD P15428 4/20 0.35
LMNA P02545 2/20 0.35
MAPK14 Q16539 2/20 0.35
AKR1B1 P15121 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29628298 0.77 TSHR (0.44) TSHRPARP1
SCHEMBL2729681 0.75 KCNJ1 (0.47) PARP1
SCHEMBL18623590 0.73 TSHR (0.47) TSHRRAB9ANPC1PARP1ALDH1A1
SCHEMBL4818156 0.71 CES1 (0.56) TSHRSRD5A1SRD5A2RAB9ANPC1
Dihydrophenanthrene SCHEMBL155991 0.71 CES1 (0.68) TSHRSRD5A1SRD5A2RAB9ANPC1
Dihydrophenanthrene SCHEMBL30297028 0.71 CES1 (0.68) TSHRSRD5A1SRD5A2RAB9ANPC1
Dihydrophenanthrene SCHEMBL29404495 0.71 CES1 (0.68) TSHRSRD5A1SRD5A2RAB9ANPC1
SCHEMBL18472563 0.70 MAPT (0.54) ALDH1A1MAPTLMNAGAA
SCHEMBL286642 0.70 MAPT (0.54) ALDH1A1MAPTLMNAGAA
SCHEMBL18472558 0.70 MAPT (0.54) ALDH1A1MAPTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5480913-A DIHYDRO-PHENANTHRENE DERIVATIVES, SIDE EFFECT REDUCTION ARCH DEVELOPMENT CORPORATION (US) 1996-01-02 US disclosed
EP-0363128-B1 ANTI-ANDROGEN COMPOUNDS ARCH DEVELOPMENT CORPORATION (US) 1993-09-01 EP disclosed
US-5208263-A Dihydrophenanthrene derivatives ARCH DEVELOPMENT CORPORATION (US) 1993-05-04 US disclosed
WO-1990003979-A2 ANTI-ANDROGEN COMPOUNDS ARCH DEVELOPMENT CORPORATION (US) 1990-04-19 WO disclosed
EP-0363128-A2 Anti-androgen compounds ARCH DEVELOPMENT CORPORATION (US) 1990-04-11 EP disclosed