SCHEMBL8952863

SCHEMBL8952863

CC(C)c1nc(-c2ccccc2)cc(-c2ccc(F)cc2)c1/C=C/C(O)CC(=O)CC(=O)O

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 5/20 0.54
ESR1 P03372 1/20 0.46
CHRM1 P11229 1/20 0.46
TBXA2R P21731 1/20 0.46
PDE4A P27815 1/20 0.46
ADRA1A P35348 1/20 0.46
ALDH1A1 P00352 1/20 0.45
CYP3A4 P08684 1/20 0.45
PDE6D O43924 1/20 0.45
NR1I2 O75469 1/20 0.45
PDE4D Q08499 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8952872 1.00 HMGCR (0.54) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9271545 0.90 HMGCR (0.51) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9271553 0.90 HMGCR (0.51) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL8953313 0.89 HMGCR (0.49) HMGCR
SCHEMBL8953297 0.89 HMGCR (0.49) HMGCR
SCHEMBL9526929 0.87 HMGCR (0.61) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9526932 0.87 HMGCR (0.61) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL8953023 0.84 HMGCR (0.53) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL8953036 0.84 HMGCR (0.53) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL10434305 0.83 HMGCR (0.53) HMGCRESR1CHRM1TBXA2RPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed
EP-0356788-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1990-03-07 EP disclosed