SCHEMBL8958971

SCHEMBL8958971

COC=C(C(=O)O)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
ALDH1A1 P00352 2/20 0.50
AKR1C3 P42330 2/20 0.49
PTGS2 P35354 1/20 0.49
AKR1C2 P52895 1/20 0.49
AKR1C1 Q04828 1/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
POLB P06746 2/20 0.49
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
BCL2L1 Q07817 1/20 0.42
BAD Q92934 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MAPK1 P28482 1/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8958964 1.00 HTT (0.50) HTTALDH1A1AKR1C3PTGS2AKR1C2
SCHEMBL7942171 1.00 HTT (0.50) HTTALDH1A1AKR1C3PTGS2AKR1C2
SCHEMBL9336389 0.84 SMN1; SMN2 (0.44) HTTALDH1A1MEN1KMT2ACES2
SCHEMBL9336394 0.84 SMN1; SMN2 (0.44) HTTALDH1A1MEN1KMT2ACES2
SCHEMBL9812652 0.83 CA1 (0.48) HTTALDH1A1PTGS2MEN1KMT2A
SCHEMBL8635962 0.83 TDP1 (0.48) HTTALDH1A1AKR1C3MEN1KMT2A
SCHEMBL8958591 0.83 TDP1 (0.48) HTTALDH1A1AKR1C3MEN1KMT2A
SCHEMBL1996920 0.82 AKR1C1 (0.53) HTTALDH1A1AKR1C3PTGS2AKR1C2
SCHEMBL2407093 0.82 AKR1C1 (0.53) HTTALDH1A1AKR1C3PTGS2AKR1C2
SCHEMBL1996915 0.82 AKR1C1 (0.53) HTTALDH1A1AKR1C3PTGS2AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519048-A 3-(indol-3-yl)-propenoic acid derivatives and pharmaceutical compositions thereof MERRELL PHARMACEUTICALS INC. (US) 1996-05-21 US disclosed