SCHEMBL8959545

SCHEMBL8959545

C[C@H](N)Cn1ccc2cc(F)c(C(F)(F)F)cc21

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 20/20 0.74
HTR2A P28223 18/20 0.74
HTR2B P41595 2/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2C9 P11712 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8959554 0.89 HTR2C (0.60) HTR2CHTR2AHTR2BCYP1A2CYP3A4
Fumaric Acid SCHEMBL8959549 0.89 HTR2C (0.60) HTR2CHTR2AHTR2BCYP1A2CYP3A4
SCHEMBL8959822 0.86 HTR2C (0.54) HTR2CHTR2AHTR2BCYP1A2CYP3A4
SCHEMBL8959826 0.86 HTR2C (0.54) HTR2CHTR2AHTR2BCYP1A2CYP3A4
SCHEMBL8959516 0.85 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2CYP3A4
SCHEMBL8959582 0.85 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2CYP3A4
SCHEMBL13970610 0.81 HTR2C (0.80) HTR2CHTR2AHTR2BCYP1A2CYP3A4
SCHEMBL8959930 0.80 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2CYP3A4
SCHEMBL8001642 0.80 HTR2C (0.78) HTR2CHTR2AHTR2BCYP1A2CYP3A4
SCHEMBL9233642 0.80 HTR2C (0.78) HTR2CHTR2AHTR2BCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN claimed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN claimed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP claimed
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP disclosed