SCHEMBL8959596

SCHEMBL8959596

CC(N)Cn1ccc2ccc(F)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 20/20 1.00
HTR2A P28223 18/20 1.00
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2C9 P11712 1/20 0.62
HTR2B P41595 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31060129 1.00 HTR2C (1.00) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959602 1.00 HTR2C (1.00) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL9229424 1.00 HTR2C (1.00) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
Fumaric Acid SCHEMBL8959564 0.88 HTR2C (0.78) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
Fumaric Acid SCHEMBL8959556 0.88 HTR2C (0.78) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959698 0.87 HTR2C (1.00) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959794 0.87 HTR2C (1.00) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL7994160 0.87 HTR2C (1.00) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL26673242 0.87 HTR2C (0.77) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959921 0.84 HTR2C (0.72) HTR2CHTR2ACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN claimed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN claimed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP claimed
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP disclosed