SCHEMBL8960046

SCHEMBL8960046

CCOC(=O)c1ccc(C#Cc2ccc(C(C)(C)CCC(C)C)cc2)nc1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.48
RARA P10276 1/20 0.48
RARB P10826 1/20 0.48
RARG P13631 1/20 0.48
KMT2A Q03164 1/20 0.48
GRM5 P41594 4/20 0.47
ACACB O00763 11/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8960507 0.85 RARB (0.55) CYP3A4RARARARBRARGKMT2A
SCHEMBL8960192 0.81 CYP3A4 (0.50) CYP3A4RARARARBRARGKMT2A
SCHEMBL9142798 0.76 CYP3A4 (0.48) CYP3A4RARARARBRARGKMT2A
SCHEMBL9142795 0.76 CYP3A4 (0.48) CYP3A4RARARARBRARGKMT2A
SCHEMBL8960230 0.75 CYP3A4 (0.52) CYP3A4RARARARBRARGKMT2A
SCHEMBL8960129 0.74 CYP3A4 (0.54) CYP3A4RARARARBRARGKMT2A
SCHEMBL5413867 0.73 CYP3A4 (0.48) CYP3A4RARARARBRARGKMT2A
SCHEMBL6411960 0.72 KMT2A (0.52) CYP3A4RARARARBRARGKMT2A
SCHEMBL9425628 0.71 RARB (0.61) CYP3A4RARBRARGKMT2AACACB
SCHEMBL6091139 0.70 KMT2A (0.49) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516904-A SKIN AND IMMUNE DISORDERS; ANTIARTHRITIC AGENTS; WOUND HEALING AGENTS ALLERGAN, INC. (US) 1996-05-14 US disclosed
EP-0436398-B1 Acetylenes disubstituted with a heteroaromatic group and a substituted phenyl group having retinoid like activity ALLERGAN INC (US) 1996-01-31 EP disclosed
US-5414007-A Skin disorders ALLERGAN, INC. (US) 1995-05-09 US disclosed
US-5264456-A Skin disorders, anticarcinogenic agents, antiarthritic agents, immunology or wound healing agents ALLERGAN, INC. (US) 1993-11-23 US disclosed
US-5175185-A Antiacne agents ALLERGAN, INC. (US) 1992-12-29 US disclosed
EP-0436398-A1 Acetylenes disubstituted with a heteroaromatic group and a substituted phenyl group having retinoid like activity ALLERGAN, INC. (US) 1991-07-10 EP disclosed
US-5013744-A Skin disorders ALLERGAN, INC. (US) 1991-05-07 US disclosed