SCHEMBL896023

SCHEMBL896023

COC(=O)N[C@@H](C(=O)N1CCC[C@H]1C(=O)Nc1ccc2[nH]c(-c3ccc(NC(=O)[C@@H]4CCCN4C(=O)[C@@H](c4ccccc4)N(C)C(=O)O)cc3)cc2c1)c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.66
CYP2C9 P11712 6/20 0.59
CYP2C19 P33261 6/20 0.59
CYP3A4 P08684 5/20 0.59
CYP2D6 P10635 2/20 0.59
CYP1A2 P05177 2/20 0.59
ALDH1A1 P00352 3/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
ROCK2 O75116 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
EP300 Q09472 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10223645 0.94 KCNH2 (0.75) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL16188305 0.91 KCNH2 (0.72) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL18379298 0.91 KCNH2 (0.72) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL20952515 0.91 KCNH2 (0.72) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL10222773 0.91 KCNH2 (0.71) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL894497 0.90 KCNH2 (0.49) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL16309220 0.90 KCNH2 (0.58) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL20952287 0.89 KCNH2 (0.56) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL16291016 0.89 KCNH2 (0.56) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL16291015 0.89 KCNH2 (0.56) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120083483-A1 INHIBITORS OF HEPATITIS C VIRUS REPLICATION MERCK SHARP & DOHME CORP (NJ) 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120083483-A1 INHIBITORS OF HEPATITIS C VIRUS REPLICATION HAVCR2, HCCS, EIF2AK2 KCNH2 4621/4885CYP2C9 2551/4885CYP2C19 3129/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.