SCHEMBL8961360

SCHEMBL8961360

CC(O)[C@H](CC(=O)O)NC(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
CA7 P43166 2/20 0.56
CYP2D6 P10635 1/20 0.50
CTSK P43235 8/20 0.44
CTSS P25774 5/20 0.44
KLK5 Q9Y337 2/20 0.43
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CA4 P22748 1/20 0.39
CA9 Q16790 1/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16970604 1.00 CA1 (0.56) CA1CA2CA7CYP2D6CTSK
SCHEMBL272148 1.00 CA1 (0.56) CA1CA2CA7CYP2D6CTSK
SCHEMBL68450 0.88 CA1 (0.67) CA1CA2CA7CYP2D6CTSK
SCHEMBL68451 0.88 CA1 (0.67) CA1CA2CA7CYP2D6CTSK
SCHEMBL969077 0.88 CA1 (0.67) CA1CA2CA7CYP2D6CTSK
SCHEMBL168390 0.85 CA1 (0.54) CA1CA2CA7CYP2D6CTSK
SCHEMBL16970732 0.85 CA1 (0.54) CA1CA2CA7CYP2D6CTSK
SCHEMBL2987820 0.83 CA1 (0.53) CA1CA2CA7CYP2D6CTSK
SCHEMBL14265317 0.83 CA1 (0.53) CA1CA2CA7CYP2D6CTSK
SCHEMBL385451 0.83 CA1 (0.53) CA1CA2CA7CYP2D6CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5480893-A ANTITUMOR MERCK & CO., INC. (US) 1996-01-02 US disclosed
US-5340828-A Anticarcinogenic agents MERCK & CO., INC. (US) 1994-08-23 US disclosed
EP-0535730-A2 Inhibitors of farnesyl protein transferase MERCK & CO. INC. (US) 1993-04-07 EP disclosed