Dimoxamine

Dimoxamine

SCHEMBL896149

CC[C@H](N)Cc1cc(OC)c(C)cc1OC

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.54
HTR2A P28223 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimoxamine SCHEMBL894999 1.00 TAAR1 (0.54) TAAR1HTR2A
Dimoxamine SCHEMBL29633087 1.00 TAAR1 (0.54) TAAR1HTR2A
Dimoxamine SCHEMBL43489 1.00 TAAR1 (0.54) TAAR1HTR2A
Dimoxamine SCHEMBL29543489 1.00 TAAR1 (0.54) TAAR1HTR2A
Dimoxamine SCHEMBL30855253 0.98 TAAR1 (0.53) TAAR1HTR2A
Dimoxamine SCHEMBL3142009 0.98 TAAR1 (0.53) TAAR1HTR2A
Dimoxamine SCHEMBL121888 0.98 TAAR1 (0.53) TAAR1HTR2A
Dimoxamine SCHEMBL30855252 0.98 TAAR1 (0.53) TAAR1HTR2A
Dimoxamine SCHEMBL3147518 0.97 TAAR1 (0.51) TAAR1HTR2A
SCHEMBL11737197 0.91 TAAR1 (0.45) TAAR1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9879293-B2 Enzymatic transamination of cyclopamine analogs INFINITY PHARMACEUTICALS, INC. (US) 2018-01-30 US disclosed
US-20160177354-A1 ENZYMATIC TRANSAMINATION OF CYCLOPAMINE ANALOGS SAFC, INC. 2016-06-23 US disclosed
EP-2462115-B1 ENZYMATIC TRANSAMINATION OF CYCLOPAMINE ANALOGS INFINITY PHARMACEUTICALS INC (US) 2016-01-06 EP disclosed
US-20140371456-A1 Enzymatic Transamination of Cyclopamine Analogs ROYALTY SECURITY, LLC 2014-12-18 US disclosed
US-8703448-B2 Enzymatic transamination of cyclopamine analogs INFINITY PHARMACEUTICALS, INC. (US) 2014-04-22 US disclosed
US-20120083607-A1 Enzymatic Transamination of Cyclopamine Analogs INFINITY PHARMACEUTICALS, INC. (US) 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120083607-A1 Enzymatic Transamination of Cyclopamine Analogs TKT, TALDO1, BCHE TAAR1 2537/4885HTR2A 4028/4885
US-20140371456-A1 Enzymatic Transamination of Cyclopamine Analogs TKT, TALDO1, BCHE TAAR1 2537/4885HTR2A 4028/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.