SCHEMBL8962829

SCHEMBL8962829

Cl/C=C/[C@H]1CC[C@H](CCC2CCC(c3ccc(Br)cc3)CC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 8/20 0.41
ESR1 P03372 6/20 0.39
CYP2C9 P11712 3/20 0.39
CYP3A4 P08684 2/20 0.39
HDAC2 Q92769 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP2D6 P10635 1/20 0.36
MAOB P27338 3/20 0.33
MAOA P21397 2/20 0.33
CCR2 P41597 1/20 0.32
DGAT1 O75907 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962823 1.00 ESR2 (0.41) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL9300179 0.91 HDAC2 (0.43) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL8962820 0.91 HDAC2 (0.43) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL8963260 0.86 CYP2C9 (0.52) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL8963140 0.86 ESR2 (0.41) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL8963133 0.86 ESR2 (0.41) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL8963099 0.86 HDAC2 (0.40) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL8963395 0.86 HDAC2 (0.40) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL8963107 0.86 HDAC2 (0.40) ESR2ESR1CYP2C9CYP3A4HDAC2
SCHEMBL8963012 0.85 ESR2 (0.41) ESR2ESR1CYP2C9CYP3A4HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed