Temiverine

Temiverine

SCHEMBL896437

CCN(CC)CC#CC(C)(C)OC(=O)[C@@](O)(c1ccccc1)C1CCCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 7/20 0.70
CHRM1 P11229 7/20 0.70
CHRM4 P08173 5/20 0.70
CHRM3 P20309 5/20 0.70
KCNH2 Q12809 3/20 0.70
CYP2C19 P33261 2/20 0.70
SLC6A3 Q01959 2/20 0.70
CYP1A2 P05177 1/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
PKM P14618 1/20 0.70
NFKB1 P19838 1/20 0.70
THPO P40225 1/20 0.70
ABCB11 O95342 1/20 0.70
ESR1 P03372 1/20 0.70
CHRM5 P08912 1/20 0.70
ADRA2A P08913 1/20 0.70
ADORA3 P0DMS8 1/20 0.70
TBXA2R P21731 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Temiverine SCHEMBL120687 1.00 CHRM2 (0.70) CHRM2CHRM1CHRM4CHRM3KCNH2
Temiverine SCHEMBL332032 0.99 MEN1 (0.71) CHRM2CHRM1CHRM4CHRM3KCNH2
Temiverine SCHEMBL6816326 0.99 CHRM2 (0.69) CHRM2CHRM1CHRM4CHRM3KCNH2
Temiverine SCHEMBL1650105 0.98 CHRM2 (0.68) CHRM2CHRM1CHRM4CHRM3KCNH2
Temiverine SCHEMBL5592324 0.98 MEN1 (0.70) CHRM2CHRM1CHRM4CHRM3KCNH2
Hydrochloric Acid SCHEMBL9878351 0.98 MEN1 (0.69) CHRM2CHRM1CHRM4CHRM3KCNH2
Hydrochloric Acid SCHEMBL9878913 0.90 POLB (0.61) CHRM2CHRM1CHRM4CHRM3KCNH2
Hydrochloric Acid SCHEMBL9878732 0.89 POLB (0.59) CHRM2CHRM1CHRM4CHRM3KCNH2
SCHEMBL7274104 0.87 CHRM2 (0.54) CHRM2CHRM1CHRM4CHRM3KCNH2
SCHEMBL9618325 0.85 POLB (0.54) CHRM2CHRM1CHRM4CHRM3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8793078-B2 Method for predicting activation energy using atomic fingerprint descriptor or atomic descriptor BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2014-07-29 US disclosed
US-20120084012-A1 METHOD FOR PREDICTING ACTIVATION ENERGY USING ATOMIC FINGERPRINT DESCRIPTOR OR ATOMIC DESCRIPTOR BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2012-04-05 US disclosed
US-20110213558-A1 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2011-09-01 US disclosed
EP-2354987-A2 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR Bioinformatics&Molecular Design Research Center (KR) 2011-08-10 EP disclosed