SCHEMBL8970541

SCHEMBL8970541

CCC(=O)OC1(c2ccccc2)CCN(CCOC(CN(C)C(=O)OCc2ccccc2)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 5/20 0.45
TACR1 P25103 3/20 0.45
DRD3 P35462 1/20 0.44
CCR5 P51681 2/20 0.41
OPRM1 P35372 2/20 0.40
OPRD1 P41143 2/20 0.40
OPRK1 P41145 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8971211 0.88 TACR2 (0.58) TACR2TACR1
SCHEMBL8969265 0.85 TACR2 (0.60) TACR2TACR1
SCHEMBL8970508 0.77 TACR2 (0.57) TACR2TACR1
SCHEMBL7312740 0.76 TACR2 (0.68) TACR2TACR1
Hydrochloric Acid SCHEMBL7745899 0.75 TACR2 (0.67) TACR2TACR1
SCHEMBL8971053 0.74 TACR2 (0.60) TACR2TACR1CCR5
SCHEMBL8973619 0.74 TACR2 (0.60) TACR2TACR1
SCHEMBL8970454 0.74 TACR2 (0.75) TACR2TACR1
SCHEMBL9119789 0.72 TACR2 (0.60) TACR2TACR1
SCHEMBL19717856 0.69 DRD3 (0.64) DRD3OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700386-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1996-03-13 EP disclosed
WO-1995026338-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1995-10-05 WO disclosed