SCHEMBL8973408

SCHEMBL8973408

N[C@]1(C(=O)O)C[C@H](C(=O)O)N(Cc2ccc(OCc3ccccc3)cc2)C1

nearest known ligand 0.78

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM6 O15303 1/20 0.78
GRM2 Q14416 7/20 0.67
GRM5 P41594 1/20 0.62
GRM3 Q14832 4/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973264 0.88 GRM6 (1.00) GRM6GRM2GRM5GRM3
SCHEMBL8061968 0.88 GRM6 (1.00) GRM6GRM2GRM5GRM3
SCHEMBL8973209 0.86 GRM6 (0.69) GRM6GRM2GRM5GRM3
SCHEMBL8973013 0.85 GRM6 (0.87) GRM6GRM2GRM5GRM3
SCHEMBL8973121 0.81 GRM6 (0.81) GRM6GRM2GRM5GRM3
SCHEMBL8973457 0.81 GRM6 (0.80) GRM6GRM2GRM5GRM3
SCHEMBL8973283 0.81 GRM2 (1.00) GRM6GRM2GRM5GRM3
SCHEMBL8973223 0.81 GRM2 (1.00) GRM6GRM2GRM5GRM3
SCHEMBL8973090 0.78 GRM6 (0.79) GRM6GRM2GRM5GRM3
SCHEMBL4663769 0.78 GRM6 (0.74) GRM6GRM2GRM5GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703218-A1 Pyrrolidinyl di-carboxylic acid derivatives as metabotropic glutamate receptor antagonists ELI LILLY AND COMPANY (US) 1996-03-27 EP disclosed
WO-1996005828-A1 PYRROLIDINYL DI-CARBOXYLIC ACID DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1996-02-29 WO disclosed