SCHEMBL8976707

SCHEMBL8976707

CCOC(=O)N1CCC(N[C@H]2CC[C@H](n3c(=O)[nH]c4ccccc43)CC2)CC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.76
CHRM2 P08172 1/20 0.76
CHRM4 P08173 1/20 0.76
CHRM5 P08912 1/20 0.76
CHRM3 P20309 1/20 0.76
ALDH1A1 P00352 3/20 0.58
MAPK1 P28482 1/20 0.55
OPRM1 P35372 2/20 0.54
HTR1A P08908 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
TACR2 P21452 1/20 0.54
DRD1 P21728 1/20 0.54
DRD5 P21918 1/20 0.54
SLC6A2 P23975 1/20 0.54
ADRA1D P25100 1/20 0.54
HTR1B P28222 1/20 0.54
TSPO P30536 1/20 0.54
ADORA1 P30542 1/20 0.54
ADRA1A P35348 1/20 0.54
ADRA1B P35368 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8976698 1.00 CHRM1 (0.76) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL4669587 0.90 CHRM1 (0.91) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL6580373 0.86 CHRM1 (1.00) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL3003287 0.82 CHRM1 (0.88) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL13243429 0.82 CHRM1 (0.88) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL13243457 0.82 CHRM1 (0.88) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL2990749 0.80 CHRM1 (0.70) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL1834035 0.79 CHRM1 (0.66) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL1837210 0.79 CHRM1 (0.69) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL3633996 0.79 CHRM1 (0.72) CHRM1CHRM2CHRM4CHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5574044-A BENZIMIDAZOL-2-ONE COMPOUNDS FOR TREATMENT OF MYOPIA MERCK & CO., INC. (US) 1996-11-12 US disclosed
WO-1996013262-A1 MUSCARINE ANTAGONISTS MERCK & CO., INC. (US) 1996-05-09 WO disclosed