SCHEMBL8989990

SCHEMBL8989990

CN(C(=O)OC(C)(C)C)C(=S)[C@@H]1CCCN1C

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
HSD11B1 P28845 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPC1 O15118 1/20 0.32
HPGD P15428 1/20 0.32
GAA P10253 1/20 0.31
CASP3 P42574 1/20 0.31
LMNA P02545 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
EPHX1 P07099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5737327 0.85 HSD17B10 (0.37) HSD17B10CYP3A4CYP2D6HSD11B1SMN1; SMN2
SCHEMBL7362291 0.75 HSD17B10 (0.42) HSD17B10CA1CA2CYP3A4CYP2D6
SCHEMBL12084380 0.75 HSD17B10 (0.42) HSD17B10CA1CA2CYP3A4CYP2D6
SCHEMBL17595517 0.70 HPGD (0.41) HSD17B10CYP3A4CYP2D6HPGDCASP3
SCHEMBL25730353 0.70 HPGD (0.41) HSD17B10CYP3A4CYP2D6HPGDCASP3
SCHEMBL17595518 0.70 HPGD (0.41) HSD17B10CYP3A4CYP2D6HPGDCASP3
SCHEMBL4590220 0.70 HSD17B10 (0.54) HSD17B10SMN1; SMN2NPC1LMNANPSR1
SCHEMBL15665375 0.69 CYP3A4 (0.43) HSD17B10CA1CA2CYP3A4CYP2D6
SCHEMBL5734517 0.69 CYP3A4 (0.43) HSD17B10CA1CA2CYP3A4CYP2D6
SCHEMBL3085529 0.69 HPGD (0.47) HSD17B10HPGDEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578633-A VASOPRESSIN AND OXYTOCIN ANTAGONISTS SANOFI (FR) 1996-11-26 US disclosed
US-5481005-A N-sulfonylindoline derivatives, their preparation and the pharmaceutical compositions in which they are present SANOFI (FR) 1996-01-02 US disclosed
US-5397801-A Affinity for vasopressin and ocytocin receptors; disorders of nervous, cardiovascular and gastrointestinal systems SANOFI (FR) 1995-03-14 US disclosed
US-5338755-A Have affinity for vasopressin and ocytocin receptors; intermediates for drugs that act on central nervous system ELF SANOFI (FR) 1994-08-16 US disclosed