SCHEMBL8993394

SCHEMBL8993394

Cc1cccc(CN2CCC(Oc3cc4cc[nH]c(=O)c4cc3C)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.53
PRKACA P17612 3/20 0.47
PRKACG P22612 3/20 0.47
PRKACB P22694 3/20 0.47
DRD4 P21917 2/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
SCN1A P35498 1/20 0.42
SCN8A Q9UQD0 1/20 0.42
ENPP2 Q13822 1/20 0.42
CHRM2 P08172 1/20 0.41
CHRM3 P20309 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8937945 0.91 ROCK1 (0.56) ROCK1PRKACAPRKACGPRKACBSCN1A
SCHEMBL8938144 0.91 MAP2K1 (0.53) ROCK1PRKACAPRKACGPRKACBBCHE
SCHEMBL8937993 0.91 ROCK1 (0.52) ROCK1PRKACAPRKACGPRKACBDRD4
SCHEMBL8937943 0.89 ROCK1 (0.56) ROCK1PRKACAPRKACGPRKACBBCHE
SCHEMBL8937944 0.88 ROCK1 (0.52) ROCK1PRKACAPRKACGPRKACBACHE
SCHEMBL8939144 0.87 ROCK1 (0.52) ROCK1PRKACAPRKACGPRKACBSCN1A
SCHEMBL8937994 0.86 ROCK1 (0.55) ROCK1PRKACAPRKACGPRKACBDRD4
SCHEMBL4006061 0.86 ROCK1 (0.56) ROCK1PRKACAPRKACGPRKACB
SCHEMBL8937973 0.86 ROCK1 (0.51) ROCK1PRKACAPRKACGPRKACBSCN1A
SCHEMBL8937933 0.85 ROCK1 (0.54) ROCK1PRKACAPRKACGPRKACBSCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed