SCHEMBL9002872

SCHEMBL9002872

CN(C)c1ccccc1CC(=O)N1C[C@@H]2[C@H](O)CCC(c3ccccc3)(c3ccccc3)[C@@H]2C1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.68
FNTA P49354 7/20 0.52
FNTB P49356 7/20 0.52
OPRD1 P41143 6/20 0.38
OPRK1 P41145 6/20 0.38
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
OPRM1 P35372 2/20 0.36
BRD4 O60885 1/20 0.35
OPRL1 P41146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9003112 1.00 TACR1 (0.68) TACR1FNTAFNTBOPRD1OPRK1
SCHEMBL9271043 1.00 TACR1 (0.68) TACR1FNTAFNTBOPRD1OPRK1
SCHEMBL9269132 0.89 TACR1 (0.59) TACR1FNTAFNTBOPRD1OPRK1
SCHEMBL9270016 0.89 TACR1 (0.59) TACR1FNTAFNTBOPRD1OPRK1
Hydrochloric Acid SCHEMBL9267078 0.88 TACR1 (0.58) TACR1FNTAFNTBOPRD1OPRK1
Hydrochloric Acid SCHEMBL9003414 0.88 TACR1 (0.58) TACR1FNTAFNTBOPRD1OPRK1
Hydrochloric Acid SCHEMBL9273776 0.88 TACR1 (0.58) TACR1FNTAFNTBOPRD1OPRK1
SCHEMBL9003093 0.84 FNTA (0.72) TACR1FNTAFNTBMEN1CYP3A4
SCHEMBL9002933 0.82 TACR1 (0.58) TACR1FNTAFNTBOPRD1OPRK1
SCHEMBL9268760 0.82 TACR1 (0.60) TACR1FNTAFNTBOPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5508433-A Derivatives of perhydroisoindole and preparation thereof RHONE-POULENC RORER S.A. (FR) 1996-04-16 US disclosed
US-5451601-A Perhydroisoindole derivatives and pharmaceutical compositions containing them RHONE-POULENC RORER S.A. (FR) 1995-09-19 US disclosed