SCHEMBL9004358

SCHEMBL9004358

CCCCC1CCC[N]C1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.56
NOS1 P29475 2/20 0.37
NOS2 P35228 2/20 0.37
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
MAPT P10636 1/20 0.31
SIGMAR1 Q99720 2/20 0.31
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7471375 0.94 CYP1A2 (0.48) CYP1A2NOS1NOS2LMNAMAPK1
SCHEMBL10377599 0.92 CYP1A2 (0.47) CYP1A2NOS1NOS2HTTSIGMAR1
SCHEMBL6399663 0.87
SCHEMBL6403085 0.87 CYP1A2 (0.67) CYP1A2NOS1NOS2LMNAMAPK1
SCHEMBL1547442 0.87
SCHEMBL8745712 0.86 CYP1A2 (0.50) CYP1A2NOS1NOS2HTTSIGMAR1
SCHEMBL6050189 0.83 CYP1A2 (0.38) CYP1A2
SCHEMBL4854731 0.81 CYP1A2 (0.41) CYP1A2NOS1NOS2
SCHEMBL2733122 0.81 CYP1A2 (0.41) CYP1A2NOS1NOS2LMNAMAPK1
SCHEMBL4536346 0.79 EPHX1 (0.41) CYP1A2HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5574037-A MODULATED BY SINO-ATRIAL NODE, ANTIISCHEMIC AGENT IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-11-12 US claimed
EP-0431856-B1 Heterocyclic compounds ZENECA LTD (GB) 1995-07-12 EP claimed
EP-0431856-A2 Heterocyclic compounds ZENECA LIMITED (GB) 1991-06-12 EP claimed
US-5574037-A MODULATED BY SINO-ATRIAL NODE, ANTIISCHEMIC AGENT IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-11-12 US disclosed
EP-0431856-B1 Heterocyclic compounds ZENECA LTD (GB) 1995-07-12 EP disclosed
US-5332737-A Cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-07-26 US disclosed
EP-0431856-A2 Heterocyclic compounds ZENECA LIMITED (GB) 1991-06-12 EP disclosed