SCHEMBL9004885

SCHEMBL9004885

CC(=O)O[C@@](Cn1cncn1)(c1ccc(Cl)cc1)[C@@H](C)n1ccnn1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.41
CYP3A4 P08684 5/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
MC4R P32245 2/20 0.35
MC3R P41968 1/20 0.35
MC1R Q01726 1/20 0.35
CYP2C9 P11712 3/20 0.34
CYP2C19 P33261 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP19A1 P11511 1/20 0.34
KCNH2 Q12809 1/20 0.33
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 1/20 0.32
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9005072 0.91 KMT2A (0.41) KMT2ACYP3A4MC3RCYP2C9CYP2C19
SCHEMBL9005114 0.81 CYP3A4 (0.34) KMT2ACYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL9005045 0.81 KMT2A (0.49) KMT2ACYP3A4ALDH1A1MAPTHTT
SCHEMBL9005065 0.78 KMT2A (0.42) KMT2ACYP3A4ALDH1A1MC3RCYP2C9
SCHEMBL9005037 0.71 KMT2A (0.49) KMT2ACYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL9005053 0.71 KMT2A (0.39) KMT2ACYP3A4ALDH1A1CYP2C9CYP2C19
SCHEMBL10434430 0.70 KMT2A (0.48) KMT2ACYP3A4ALDH1A1MAPTHTT
SCHEMBL9004935 0.69 CYP3A4 (0.40) KMT2ACYP3A4ALDH1A1CYP2C9CYP2C19
SCHEMBL9835984 0.69 KMT2A (0.46) KMT2ACYP3A4ALDH1A1MAPTHTT
SCHEMBL9844009 0.68 KMT2A (0.48) KMT2ACYP3A4ALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495024-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 1996-02-27 US disclosed
US-5371100-A An 1-(1H-1,2,4-triazolyl) or 1-(1H-imidazolyl)-2-phenyl-3-(1H or 2H-tetrazolyl)-2-alkylol or alkyloxyacetyl fungicides for fungal infections TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-06 US disclosed
EP-0548553-A1 Optically active azole compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-06-30 EP disclosed