SCHEMBL9006953

SCHEMBL9006953

C#Cc1ccc2c(c1)OC(C)(C)CC2(C)C

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.31
CYP26A1 O43174 1/20 0.31
CYP26B1 Q9NR63 1/20 0.31
FTO Q9C0B1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5736909 0.87 AKR1B1 (0.35) AKR1B1CYP26A1CYP26B1FTO
SCHEMBL9006905 0.80 AKR1B1 (0.32) AKR1B1CYP26A1FTO
SCHEMBL7218162 0.76 CYP26A1 (0.42) AKR1B1CYP26A1CYP26B1FTO
SCHEMBL9484220 0.75 RARB (0.41) CYP26A1
SCHEMBL9007036 0.75 RARB (0.60) CYP26A1
SCHEMBL9054386 0.75 MAPT (0.42) AKR1B1CYP26A1CYP26B1FTO
SCHEMBL8759623 0.75 BACE1 (0.42) AKR1B1CYP26A1CYP26B1FTO
SCHEMBL8561808 0.73 AKR1B1 (0.33) AKR1B1CYP26A1CYP26B1FTO
SCHEMBL5735185 0.72
SCHEMBL9007040 0.71 AKR1B1 (0.36) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0571546-B1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN INC (US) 1996-10-16 EP disclosed
US-5346915-A Chromans and thiochromans with phenylethynyl substituents at the 7-position having retinold-like biological activity ALLERGAN, INC. (US) 1994-09-13 US disclosed
US-5346895-A Treating dermatoses, immunological disorders, wound healing ALLERGAN, INC. (US) 1994-09-13 US disclosed
EP-0577737-A1 CHROMANS AND THIOCHROMANS WITH HETEROARYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 1994-01-12 EP disclosed
WO-1992017471-A1 CHROMANS AND THIOCHROMANS WITH HETEROARYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 1992-10-15 WO disclosed