SCHEMBL9007565

SCHEMBL9007565

O=Cc1ccc2c(Br)c(O)ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.53
ESR2 Q92731 3/20 0.53
KDM4E B2RXH2 1/20 0.52
PTGS2 P35354 1/20 0.52
RAB9A P51151 1/20 0.52
ERN1 O75460 7/20 0.51
HSD17B1 P14061 1/20 0.49
HSD17B2 P37059 1/20 0.49
POLB P06746 1/20 0.48
ALDH1A1 P00352 4/20 0.43
ALDH5A1 P51649 3/20 0.43
ABAT P80404 3/20 0.43
TRIM24 O15164 1/20 0.43
HPGD P15428 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TRIM33 Q9UPN9 1/20 0.43
AOX1 Q06278 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10331755 0.81 KDM4E (0.55) ESR1ESR2KDM4EPTGS2RAB9A
SCHEMBL4362335 0.79 ESR1 (0.53) ESR1ESR2KDM4EPTGS2RAB9A
SCHEMBL18998873 0.79 KDM4E (0.52) ESR1ESR2KDM4EPTGS2RAB9A
SCHEMBL10827942 0.79 ESR1 (0.54) ESR1ESR2KDM4EPTGS2RAB9A
SCHEMBL4358501 0.79 ESR1 (0.53) ESR1ESR2KDM4EPTGS2RAB9A
SCHEMBL9127399 0.78 CYP2A6 (0.48) KDM4EPTGS2RAB9AERN1ALDH1A1
SCHEMBL11809502 0.76 ERN1 (0.56) KDM4EPTGS2RAB9AERN1ALDH1A1
SCHEMBL9623620 0.75 ESR1 (0.72) ESR1ESR2ERN1HSD17B1HSD17B2
SCHEMBL50832 0.75 ESR1 (0.61) ESR1ESR2KDM4EERN1HSD17B1
SCHEMBL30570998 0.75 ESR1 (0.72) ESR1ESR2ERN1HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5482968-A ENZYME INHIBITORS, HYPOGLYCEMIC AGENTS AND VASCULAR AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1996-01-09 US disclosed
US-5399588-A Diabetes treatment AMERICAN HOME PRODUCTS CORPORATION (US) 1995-03-21 US disclosed