SCHEMBL9010860

SCHEMBL9010860

O=C(S)C1c2ccccc2-c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.57
HDAC4 P56524 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
HDAC9 Q9UKV0 1/20 0.57
HDAC5 Q9UQL6 1/20 0.57
NCOR2 Q9Y618 1/20 0.57
POLB P06746 1/20 0.45
KMT2A Q03164 2/20 0.41
HBB P68871 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TSHR P16473 2/20 0.40
CYP1A2 P05177 1/20 0.40
EDNRB P24530 1/20 0.39
EDNRA P25101 1/20 0.39
MAPT P10636 2/20 0.39
GPR3 P46089 1/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30001332 0.78 HDAC3 (0.59) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL40500 0.78 HDAC3 (0.59) HDAC3HDAC4HDAC7HDAC8HDAC6
Benzene SCHEMBL28538497 0.78 HDAC3 (0.59) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL1567079 0.78 HDAC3 (0.59) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL7043488 0.76 HDAC3 (0.57) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL30250175 0.76 ATM (0.61) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL3143561 0.76 ATM (0.61) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL4796539 0.76 HDAC3 (0.57) HDAC3HDAC4HDAC7HDAC8HDAC6
SCHEMBL15125189 0.76 HDAC3 (0.57) HDAC3HDAC4HDAC7HDAC8HDAC6
Hydrochloric Acid SCHEMBL7052205 0.76 HDAC3 (0.57) HDAC3HDAC4HDAC7HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0542392-B1 Use of thiol-S-(2-diethyl-aminoethyl)-ester compound for the preparation of a medicament for the treating neuro-muscular incontinence UNITED PHARMACEUTICALS INC (US) 1996-11-13 EP disclosed
EP-0542392-A1 Use of thiol-S-(2-diethyl-aminoethyl)-ester compound for the preparation of a medicament for the treating neuro-muscular incontinence United Pharmaceuticals, Inc. (US) 1993-05-19 EP disclosed
US-5130336-A Administering a thiol-dimethylaminoethyl ester compound UNITED PHARMACEUTICALS, INC. (US) 1992-07-14 US disclosed
US-RE33907-E Anti-spasmodic agents having a heterocyclic ring UNITED PHARMACEUTICALS, INC. (US) 1992-04-28 US disclosed
US-4957941-A Anti-spasmdoic agents having an acetylenic bond UNITED PHARMACEUTICALS, INC. (US) 1990-09-18 US disclosed
US-4918082-A Anti-spasmodic agents containing quaternary nitrogen UNITED PHARMACEUTICALS, INC. (US) 1990-04-17 US disclosed
US-4857535-A THIOESTERS UNITED PHARMACEUTICALS (US) 1989-08-15 US disclosed
US-4766119-A SMOOTH MUSCLE RELAXANTS UNITED PHARMACEUTICALS, INC. (US) 1988-08-23 US disclosed
EP-0267319-A1 Anti-spasmodic agents having a ring in the main chain United Pharmaceuticals, Inc. (US) 1988-05-18 EP disclosed
US-4725593-A Method of treating smooth muscle spasm UNITED PHARMACEUTICALS, INC. (US) 1988-02-16 US disclosed
US-4721783-A SMOOTH MUSCLES UNITED PHARMACEUTICALS, INC. (US) 1988-01-26 US disclosed
US-4721722-A Anti-spasmodic agents containing quaternary nitrogen UNITED PHARMACEUTICALS, INC. (US) 1988-01-26 US disclosed
US-4678780-A SMOOTH MUSCLE RELAXANTS UNITED PHARMACEUTICALS, INC. (US) 1987-07-07 US disclosed
US-4652649-A BENZOYL-THIO-S-AMINOALKYLS UNITED PHARMACEUTICALS, INC. (US) 1987-03-24 US disclosed
US-4647562-A Anti-spasmodic agents having three branch chains UNITED PHARMACEUTICALS, INC. (US) 1987-03-03 US disclosed