SCHEMBL901500

SCHEMBL901500

CCCCOC(=O)NCCCCC(=O)OCc1cc(F)c(F)cc1-c1ccc2nc(N)nc(C(=O)N3Cc4ccccc4C3)c2c1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.54
HSP90AB1 P08238 3/20 0.44
NAMPT P43490 3/20 0.38
AGTR1 P30556 2/20 0.34
AGTR2 P50052 2/20 0.34
PREP P48147 2/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP7 Q9UHL4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL901729 0.90 HSP90AA1 (0.54) HSP90AA1HSP90AB1NAMPTPREP
SCHEMBL904085 0.88 HSP90AA1 (0.56) HSP90AA1HSP90AB1NAMPT
Hydrochloric Acid SCHEMBL15091355 0.86 HSP90AA1 (0.63) HSP90AA1HSP90AB1NAMPTDPP8DPP7
SCHEMBL902377 0.86 HSP90AA1 (0.63) HSP90AA1HSP90AB1NAMPTDPP8DPP7
SCHEMBL10255169 0.86 HSP90AA1 (0.65) HSP90AA1HSP90AB1NAMPTDPP8DPP7
SCHEMBL901832 0.86 HSP90AA1 (0.64) HSP90AA1HSP90AB1NAMPT
Hydrochloric Acid SCHEMBL15091340 0.86 HSP90AA1 (0.62) HSP90AA1HSP90AB1NAMPTDPP8DPP7
Hydrochloric Acid SCHEMBL15091335 0.85 HSP90AA1 (0.64) HSP90AA1HSP90AB1NAMPT
SCHEMBL904227 0.85 HSP90AA1 (0.64) HSP90AA1HSP90AB1PREPDPP8DPP7
SCHEMBL902181 0.85 HSP90AA1 (0.57) HSP90AA1HSP90AB1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2621919-A1 PHENYLQUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2013-08-07 EP disclosed
WO-2012041435-A1 PHENYLQUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2012-04-05 WO disclosed