SCHEMBL9021645

SCHEMBL9021645

CCc1ccc(Nc2nc(N)c3ncn([C@@H]4O[C@H](CO)C(O)C4O)c3n2)cc1

nearest known ligand 0.79

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.79
CYP1A2 P05177 2/20 0.79
ADORA2B P29275 2/20 0.79
THPO P40225 1/20 0.79
MEN1 O00255 1/20 0.79
CYP2D6 P10635 1/20 0.79
CYP2C9 P11712 1/20 0.79
CYP2C19 P33261 1/20 0.79
KMT2A Q03164 1/20 0.79
BLM P54132 1/20 0.79
ADORA3 P0DMS8 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9021625 1.00 ADORA2A (0.79) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL9022416 0.93 ADORA2A (0.77) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL9022429 0.93 ADORA2A (0.77) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL9021921 0.91 ADORA2A (0.74) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL7856570 0.91 ADORA2A (0.74) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL9021901 0.91 ADORA2A (0.74) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL29753859 0.89 CYP1A2 (1.00) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL725689 0.89 CYP1A2 (1.00) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL29387702 0.89 CYP1A2 (1.00) ADORA2ACYP1A2ADORA2BTHPOMEN1
SCHEMBL725690 0.89 CYP1A2 (1.00) ADORA2ACYP1A2ADORA2BTHPOMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0704215-A2 Inhibitor of vascular permeability enhancer TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-03 EP disclosed