SCHEMBL9027700

SCHEMBL9027700

COc1ccc(C=C(C#N)C(N)=O)c2cccnc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.55
CYP2C9 P11712 2/20 0.55
CYP3A4 P08684 1/20 0.55
KDM4E B2RXH2 8/20 0.54
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
MAPT P10636 4/20 0.48
MAPK1 P28482 1/20 0.48
NEK2 P51955 3/20 0.45
PLK1 P53350 2/20 0.45
EGFR P00533 1/20 0.45
ERBB2 P04626 1/20 0.45
LMNA P02545 2/20 0.44
PKM P14618 1/20 0.44
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
ALDH1A1 P00352 3/20 0.42
POLB P06746 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7466256 0.83 KDM4E (0.56) CYP1A2CYP2C9KDM4EKMT2AMEN1
SCHEMBL8830493 0.83 KDM4E (0.56) CYP1A2CYP2C9KDM4EKMT2AMEN1
SCHEMBL7466251 0.83 KDM4E (0.56) CYP1A2CYP2C9KDM4EKMT2AMEN1
SCHEMBL28436908 0.74 KDM4E (0.76) CYP1A2CYP2C9CYP3A4KDM4EKMT2A
SCHEMBL3156151 0.74 KMT2A (0.59) KDM4EKMT2AMEN1PDE4APDE4B
SCHEMBL1388456 0.74 MCL1 (0.51) CYP1A2CYP2C9CYP3A4KDM4EKMT2A
SCHEMBL1388454 0.74 MCL1 (0.51) CYP1A2CYP2C9CYP3A4KDM4EKMT2A
SCHEMBL7471065 0.74 MCL1 (0.51) CYP1A2CYP2C9CYP3A4KDM4EKMT2A
SCHEMBL28056488 0.72 KDM4E (0.57) KDM4EKMT2AMEN1MAPTEGFR
SCHEMBL28440427 0.71 TP53 (0.67) CYP1A2CYP2C9CYP3A4KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558950-B1 3-aryl-glycidic ester derivatives and process for their preparation PHARMACIA SPA (IT) 1996-12-04 EP disclosed
US-5436235-A 3-aryl-glycidic ester derivatives FARMITALIA CARLO ERBA S.R.L. (IT) 1995-07-25 US disclosed
EP-0558950-A1 3-aryl-glycidic ester derivatives and process for their preparation PHARMACIA S.p.A. (IT) 1993-09-08 EP disclosed