SCHEMBL9028244

SCHEMBL9028244

OCCC1(c2ccc(C(F)(F)F)c(C(F)(F)F)c2)CCCCNC1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 18/20 0.64
SLC6A2 P23975 13/20 0.64
SLC6A3 Q01959 12/20 0.64
CYP2D6 P10635 4/20 0.64
TACR1 P25103 5/20 0.42
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026665 0.96 SLC6A4 (0.63) SLC6A4SLC6A2SLC6A3CYP2D6TACR1
SCHEMBL8885644 0.91 SLC6A2 (0.52) SLC6A4SLC6A2SLC6A3CYP2D6TACR1
SCHEMBL9027921 0.88 SLC6A4 (0.67) SLC6A4SLC6A2SLC6A3CYP2D6TACR1
SCHEMBL9028250 0.86 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3CYP2D6TACR1
SCHEMBL9028807 0.84 SLC6A4 (0.67) SLC6A4SLC6A2SLC6A3CYP2D6TACR1
SCHEMBL9026645 0.81 SLC6A4 (0.68) SLC6A4SLC6A2SLC6A3CYP2D6TACR1
SCHEMBL8458076 0.78 SLC6A4 (1.00) SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL9027453 0.78 SLC6A4 (0.68) SLC6A4SLC6A2SLC6A3CYP2D6TACR1
SCHEMBL8881940 0.78 SLC6A2 (0.55) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL9028214 0.76 SLC6A4 (0.67) SLC6A4SLC6A2SLC6A3CYP2D6TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed