SCHEMBL9028482

SCHEMBL9028482

CC(C)Oc1cccc(CC(=O)N2CCCC(CCN3CCN(C4CCCCC4)CC3)(c3ccc(Cl)c(Cl)c3)C2)c1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.65
TACR2 P21452 1/20 0.65
CCR5 P51681 1/20 0.52
HRH1 P35367 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9032557 1.00 TACR1 (0.65) TACR1TACR2CCR5HRH1
SCHEMBL9028476 1.00 TACR1 (0.65) TACR1TACR2CCR5HRH1
SCHEMBL9028201 0.98 TACR1 (0.64) TACR1TACR2CCR5HRH1
SCHEMBL9027621 0.98 TACR1 (0.64) TACR1TACR2CCR5HRH1
SCHEMBL8882971 0.96 TACR2 (0.70) TACR1TACR2HRH1
SCHEMBL8883494 0.96 TACR2 (0.70) TACR1TACR2HRH1
SCHEMBL8882965 0.96 TACR2 (0.70) TACR1TACR2HRH1
SCHEMBL9027942 0.94 TACR1 (0.65) TACR1TACR2CCR5HRH1
SCHEMBL9027933 0.94 TACR1 (0.65) TACR1TACR2CCR5HRH1
SCHEMBL9028136 0.93 TACR1 (0.65) TACR1TACR2CCR5HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed