SCHEMBL9028577

SCHEMBL9028577

COc1ccccc1C(=O)N1CCCC[C@](CCOS(C)(=O)=O)(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 14/20 0.58
TACR1 P25103 13/20 0.58
TACR3 P29371 4/20 0.45
HRH1 P35367 1/20 0.45
HTT P42858 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6948617 0.97 TACR2 (0.59) TACR2TACR1TACR3HRH1HTT
SCHEMBL8810091 0.94 TACR2 (0.65) TACR2TACR1TACR3HRH1
SCHEMBL8886812 0.94 TACR2 (0.65) TACR2TACR1TACR3HRH1
SCHEMBL9027948 0.91 TACR2 (0.49) TACR2TACR1HTTCYP3A4CYP2C9
SCHEMBL9028251 0.90 TACR2 (0.57) TACR2TACR1TACR3HRH1HTT
SCHEMBL9027885 0.87 TACR2 (0.58) TACR2TACR1TACR3HRH1
SCHEMBL9027870 0.86 TACR2 (0.56) TACR2TACR1TACR3HRH1
SCHEMBL6956796 0.86 TACR2 (0.63) TACR2TACR1TACR3HRH1HTT
SCHEMBL8883701 0.85 TACR2 (0.55) TACR2TACR1TACR3HRH1HTT
SCHEMBL9027802 0.85 TACR2 (0.59) TACR2TACR1TACR3HRH1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed