SCHEMBL9028985

SCHEMBL9028985

CCOc1ccc([C@@]2(CCN3CCN(C4CCCCC4)CC3)CCCCN(C(=O)Cc3cccc(OC(C)C)c3)C2)cc1OCC

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.51
TACR2 P21452 1/20 0.51
HRH1 P35367 1/20 0.44
CCR5 P51681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9028578 0.98 TACR1 (0.52) TACR1TACR2HRH1CCR5
SCHEMBL9028591 0.98 TACR1 (0.52) TACR1TACR2HRH1CCR5
SCHEMBL8882524 0.96 TACR1 (0.56) TACR1TACR2HRH1
SCHEMBL8882519 0.96 TACR1 (0.56) TACR1TACR2HRH1
SCHEMBL9028431 0.95 TACR1 (0.52) TACR1TACR2HRH1CCR5
SCHEMBL9027821 0.94 TACR1 (0.52) TACR1TACR2HRH1CCR5
SCHEMBL9027831 0.94 TACR1 (0.52) TACR1TACR2HRH1CCR5
SCHEMBL8882942 0.92 TACR1 (0.56) TACR1TACR2HRH1CCR5
SCHEMBL8882935 0.92 TACR1 (0.56) TACR1TACR2HRH1CCR5
SCHEMBL9027391 0.92 TACR1 (0.54) TACR1TACR2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563133-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1996-10-08 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed