SCHEMBL9030675

SCHEMBL9030675

CCCn1c(=O)n2c(-c3ccc([N+](=O)[O-])cc3)nnc2c2c1ncn2C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.48
PDE4A P27815 7/20 0.48
PDE4B Q07343 7/20 0.48
PDE4C Q08493 7/20 0.48
PDE4D Q08499 7/20 0.48
ADORA2B P29275 6/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TNF P01375 1/20 0.40
APOBEC3G Q9HC16 2/20 0.40
LMNA P02545 1/20 0.40
GLA P06280 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9031302 0.87 ADORA2A (0.54) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9032358 0.86 ADORA2A (0.56) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9031011 0.85 ADORA2A (0.52) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9030428 0.85 ADORA2A (0.52) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9031357 0.84 PDE4A (0.53) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9031411 0.83 PDE4A (0.50) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9031456 0.83 ADORA2A (0.50) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9032303 0.82 ADORA2A (0.54) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9031860 0.82 ADORA2A (0.49) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9031868 0.80 PDE4A (0.49) ADORA2APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP disclosed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US disclosed
EP-0417790-A2 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-20 EP disclosed