SCHEMBL9032255

SCHEMBL9032255

CCCn1c(=O)n2c(-c3cc(Cl)ccc3Cl)nnc2c2c1ncn2C

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.48
PDE4B Q07343 8/20 0.48
PDE4C Q08493 8/20 0.48
PDE4D Q08499 8/20 0.48
ADORA2A P29274 7/20 0.48
ADORA2B P29275 3/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PDE2A O00408 5/20 0.42
PDE10A Q9Y233 2/20 0.42
TNF P01375 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9031355 0.87 ADORA2A (0.50) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031011 0.85 ADORA2A (0.52) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031868 0.84 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031727 0.84 ADORA2A (0.49) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9032358 0.79 ADORA2A (0.56) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9033223 0.79 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9032171 0.79 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031302 0.78 ADORA2A (0.54) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9032369 0.77 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9031357 0.77 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP disclosed
EP-0417790-A2 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-20 EP disclosed