SCHEMBL903680

SCHEMBL903680

c1ccc([C@H]2Oc3cc(-c4cnc([C@@H]5CCCN5)[nH]4)ccc3-c3cc4cc(-c5cnc([C@@H]6CCCN6)[nH]5)ccc4n32)cc1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.32
HPGDS O60760 1/20 0.32
SSTR3 P32745 1/20 0.31
MAPK13 O15264 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30
PRCP P42785 1/20 0.30
PYGL P06737 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19225801 1.00 NR1H4 (0.32) NR1H4HPGDSSSTR3MAPK13MAPK12
SCHEMBL18978473 1.00 NR1H4 (0.32) NR1H4HPGDSSSTR3MAPK13MAPK12
SCHEMBL10215164 1.00 NR1H4 (0.32) NR1H4HPGDSSSTR3MAPK13MAPK12
SCHEMBL18057078 1.00 NR1H4 (0.32) NR1H4HPGDSSSTR3MAPK13MAPK12
SCHEMBL903494 1.00 NR1H4 (0.32) NR1H4HPGDSSSTR3MAPK13MAPK12
SCHEMBL19225806 1.00 NR1H4 (0.32) NR1H4HPGDSSSTR3MAPK13MAPK12
SCHEMBL18057083 1.00 NR1H4 (0.32) NR1H4HPGDSSSTR3MAPK13MAPK12
SCHEMBL10219365 0.94 PRCP (0.33) NR1H4HPGDSPRCP
SCHEMBL10219362 0.94 CDC7 (0.34) SSTR3PRCP
SCHEMBL18978436 0.89

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041014-A1 TETRACYCLIC INDOLE DERIVATIVES FOR TREATING HEPATITIS C VIRUS INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed