SCHEMBL9040804

SCHEMBL9040804

COC(=O)C(=C(C)c1ccccc1)c1ccccc1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.47
ALDH1A1 P00352 5/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 2/20 0.44
HPGD P15428 3/20 0.44
KDM4E B2RXH2 2/20 0.44
HSD17B10 Q99714 2/20 0.44
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
MAPT P10636 2/20 0.43
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ESR1 P03372 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
HMGB1 P09429 1/20 0.42
GGT1 P19440 1/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
BLM P54132 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9141882 1.00 AKR1C3 (0.47) AKR1C3ALDH1A1ALOX15TSHRHPGD
SCHEMBL9142024 0.91 AKR1C3 (0.55) AKR1C3ALDH1A1ALOX15HPGDKDM4E
SCHEMBL9041393 0.91 AKR1C3 (0.55) AKR1C3ALDH1A1ALOX15HPGDKDM4E
SCHEMBL9043213 0.85 AKR1C3 (0.48) AKR1C3ALDH1A1ALOX15TSHRHPGD
SCHEMBL4957182 0.84 TSHR (0.52) ALOX15TSHRHPGDKDM4EKMT2A
SCHEMBL9079039 0.78 AKR1C3 (0.42) AKR1C3ALDH1A1ALOX15TSHRHPGD
SCHEMBL9143547 0.78 AKR1C3 (0.42) AKR1C3ALDH1A1ALOX15TSHRHPGD
SCHEMBL15081529 0.76 TSHR (0.56) ALDH1A1ALOX15TSHRHPGDKDM4E
SCHEMBL14868118 0.76 TSHR (0.56) ALDH1A1ALOX15TSHRHPGDKDM4E
SCHEMBL14868116 0.76 TSHR (0.56) ALDH1A1ALOX15TSHRHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585382-A ANTICARCINOGENIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-17 US disclosed
EP-0705250-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-04-10 EP disclosed
US-5416089-A Antitumor agent THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-16 US disclosed
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed